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Therapeutic utility of cannabinoid receptor type 2 (CB(2)) selective agonists.
Cell Chem Biol 56: 8224-56 (2013)
Arena Pharmaceuticals
Discovery and optimization of piperidyl-1,2,3-triazole ureas as potent, selective, and in vivo-active inhibitors of a/ß-hydrolase domain containing 6 (ABHD6).
Cell Chem Biol 56: 8270-9 (2013)
The Scripps Research Institute
Fragment-to-hit-to-lead discovery of a novel pyridylurea scaffold of ATP competitive dual targeting type II topoisomerase inhibiting antibacterial agents.
Cell Chem Biol 56: 8712-35 (2013)
Astrazeneca R&D Boston